Testsealabs OXY Oxycodone Test
I-Oxycodone: Ulwazi Olubalulekile
I-Oxycodone iyi-opioid enga-synthetic enokufana kwesakhiwo ne-codeine. Ikhiqizwa ngokushintsha i-thebaine, i-alkaloid etholakala ku-opium poppy.
Njengawo wonke ama-opiate agonists, i-oxycodone inikeza ukukhululeka kobuhlungu ngokusebenza kuma-opioid receptors entanjeni yomgogodla, ebuchosheni, futhi ngokunokwenzeka ngqo ezicutshini ezithintekile. Inqunyelwe ukukhulula ubuhlungu obuphakathi kuya phezulu ngaphansi kwamagama okuhweba aziwayo, okuhlanganisa:
I-OxyContin®
I-Tylox®
I-Percodan®
I-Percocet®
Ngokuphawulekayo, i-Tylox®, i-Percodan®, ne-Percocet® iqukethe imithamo emincane ye-oxycodone hydrochloride ehlanganiswe namanye ama-analgesics (isb, i-acetaminophen noma i-aspirin), kuyilapho i-OxyContin® iqukethe kuphela i-oxycodone hydrochloride efomini lokukhishwa kwesikhathi.
I-Oxycodone imetabolis nge-demethylation ibe i-oxymorphone ne-noroxycodone. Ngomthamo owodwa womlomo ongu-5mg, u-33–61% ukhishwa ngomchamo wamahora angu-24, okuhlanganisa:
Isidakamizwa esingashintshiwe (13–19%)
Isidakamizwa esihlanganisiwe (7–29%)
I-oxymorphone ehlanganisiwe (13–14%)
Iwindi lokutholwa kwe-oxycodone emchameni kulindeleke ukuthi lifane nelamanye ama-opioid (isb, i-morphine).
Ukuhlolwa kwe-OXY Oxycodone kuveza umphumela omuhle lapho amazinga e-oxycodone omchamo edlula u-100 ng/mL. Okwamanje, Ukuphathwa Kwezidakamizwa Nokuphathwa Kwezinsizakalo Zezempilo Yengqondo (SAMHSA) ayikasunguli ukunqanyulwa okunconyiwe kokuhlolwa kwezibonelo ezine-oxycodone-positive.

