Testsealabs PGB Pregabalin Test
I-Pregabalin, i-analogue ye-gamma-aminobutyric acid evimbela neurotransmitter kanye ne-gabapentin, isetshenziswe emtholampilo kusukela ngo-2002 njenge-analgesic, i-anticonvulsant, ne-anxiolytic agent.
Inikezwa njengomuthi wamahhala kuma-capsules angama-25-300 mg wokuphathwa ngomlomo. Imithamo yabantu abadala ivamise ukuba phakathi kwebanga lama-50-200 mg kathathu ngosuku.
Umthamo owodwa obhalwe ngomlomo we-pregabalin kubantu wakhishwa emchamweni (92%) nasendle (<0.1%) esikhathini esiyizinsuku ezi-4. Imikhiqizo yokukhishwa komchamo yayihlanganisa izidakamizwa ezingashintshiwe (90% yomthamo), i-N-Methylpregabalin (0.9%), nezinye.
Imithamo yomlomo eyodwa engu-75 noma engu-150 mg enikezwe abantu abanempilo iveze ukugxila kwe-pregabalin ephezulu yomchamo ongu-151 noma 214 μg/mL, ngokulandelana, esibonelweni sokuqala samahora angu-8.
Amazinga omchamo we-Pregabalin kuma-specimens angu-57,542 avela ezigulini ezinobuhlungu obungapheli alinganiselwa ku-184 μg/mL.
Ukuhlolwa kwe-PGB Pregabalin kuveza umphumela omuhle lapho izinga le-pregabalin emchameni lidlula u-2,000 ng/mL.

