Testsealabs PGB Pregabalin Hoao
ʻO Pregabalin, kahi analog o ka inhibitory neurotransmitter gamma-aminobutyric acid a me ka gabapentin, ua hoʻohana ʻia i ka maʻi mai 2002 ma ke ʻano he analgesic, anticonvulsant, a me anxiolytic agent.
Hāʻawi ʻia ʻo ia ma ke ʻano he lāʻau manuahi i 25-300 mg capsules no ka hoʻokele waha. ʻO ka maʻamau o ka nui o nā pākeke he 50-200 mg ʻekolu mau lā i kēlā me kēia lā.
Hoʻopau ʻia kahi maʻi waha o pregabalin i loko o ke kanaka i loko o ka mimi (92%) a me nā feces (<0.1%) ma kahi o 4 mau lā. ʻO nā huahana urinary excretion ka lāʻau i hoʻololi ʻole ʻia (90% o ka dose), N-Methylpregabalin (0.9%), a me nā mea ʻē aʻe.
Hoʻokahi waha waha 75 a i ʻole 150 mg i hāʻawi ʻia i nā kānaka olakino i hāʻawi ʻia ka kiʻekiʻe o ka urinary pregabalin concentrations o 151 a i ʻole 214 μg/mL, i loko o ka hōʻike mua 8-hola.
Pregabalin urine pae ma 57,542 specimens mai ka maʻi maʻi eha maʻi awelika 184 μg/mL.
Hāʻawi ka PGB Pregabalin Test i kahi hopena maikaʻi ke ʻoi aku ka pae pregabalin i ka mimi ma mua o 2,000 ng/mL.

