Ikizamini cya PGB Ikizamini cya Pregabalin

Ibisobanuro bigufi:

Ikizamini cya PGB Pregabalin ni uruhande rwa chromatografique immunoassay kugirango tumenye neza pregabalin mu nkari.
gouIbisubizo Byihuse: Laboratoire-Nukuri muminota gouLaboratoire-Icyiciro Cyuzuye: Yizewe & Yizewe
gouIkizamini Ahantu hose: Nta laboratoire isabwa  gouUbwiza bwemewe: 13485, CE, Mdsap Yubahiriza
gouByoroheje & Byoroheje: Byoroshye-Gukoresha, Zeru Hassle  gouAmahirwe meza: Gerageza neza murugo

Ibicuruzwa birambuye

Ibicuruzwa

Ibiyobyabwenge byo gukoresha nabi Ikizamini cyihuse (1)
Ikizamini cya Pregabalin

Pregabalin, ikigereranyo cya inhibitori ya neurotransmitter gamma-aminobutyric ndetse na gabapentin, yakoreshejwe mubuvuzi kuva 2002 nk'umuti udakira, anticonvulsant, na anxiolytique.

Itangwa nkibiyobyabwenge byubusa muri 25-300 mg capsules yo kuyobora umunwa. Ingano yabantu bakuru mubisanzwe iri hagati ya 50-200 mg gatatu kumunsi.

 

Umunwa umwe wanditseho urugero rwa pregabalin mu bantu wakuweho mu nkari (92%) no mu mwanda (<0.1%) mugihe cyiminsi 4. Ibicuruzwa biva mu nkari birimo imiti idahindutse (90% ya dose), N-Methylpregabalin (0.9%), nibindi.

 

Indwara imwe yo mu kanwa 75 cyangwa 150 mg ihabwa abantu bazima byatanze urugero rwinkari za pregabalin zingana na 151 cyangwa 214 μg / mL, mugihe cyamasaha 8 yambere.

 

Urwego rwinkari za Pregabalin mubigereranyo 57.542 byabarwayi bafite ububabare budakira bagereranije 184 μg / mL.

 

Ikizamini cya PGB Pregabalin gitanga umusaruro ushimishije mugihe urugero rwa pregabalin mu nkari rurenze 2000 ng / mL.
Ibiyobyabwenge byo gukoresha nabi Ikizamini cyihuse (2)
Ibiyobyabwenge byo gukoresha nabi Ikizamini cyihuse (2)
Ibiyobyabwenge byo gukoresha nabi Ikizamini cyihuse (1)

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