Ikizamini cya PGB Ikizamini cya Pregabalin
Pregabalin, ikigereranyo cya inhibitori ya neurotransmitter gamma-aminobutyric ndetse na gabapentin, yakoreshejwe mubuvuzi kuva 2002 nk'umuti udakira, anticonvulsant, na anxiolytique.
Itangwa nkibiyobyabwenge byubusa muri 25-300 mg capsules yo kuyobora umunwa. Ingano yabantu bakuru mubisanzwe iri hagati ya 50-200 mg gatatu kumunsi.
Umunwa umwe wanditseho urugero rwa pregabalin mu bantu wakuweho mu nkari (92%) no mu mwanda (<0.1%) mugihe cyiminsi 4. Ibicuruzwa biva mu nkari birimo imiti idahindutse (90% ya dose), N-Methylpregabalin (0.9%), nibindi.
Indwara imwe yo mu kanwa 75 cyangwa 150 mg ihabwa abantu bazima byatanze urugero rwinkari za pregabalin zingana na 151 cyangwa 214 μg / mL, mugihe cyamasaha 8 yambere.
Urwego rwinkari za Pregabalin mubigereranyo 57.542 byabarwayi bafite ububabare budakira bagereranije 184 μg / mL.
Ikizamini cya PGB Pregabalin gitanga umusaruro ushimishije mugihe urugero rwa pregabalin mu nkari rurenze 2000 ng / mL.

