Testsealabs PGB Pregabalin Muedzo
Pregabalin, analog ye inhibitory neurotransmitter gamma-aminobutyric acid uyewo yegabapentin, yakashandiswa pakiriniki kubvira 2002 seanorapisa marwadzo, anticonvulsant, uye anxiolytic agent.
Inopihwa semushonga wemahara mu 25-300 mg capsules yekutonga nemuromo. Mishonga yevakuru inowanzova mukati mehuwandu hwe50-200 mg katatu pazuva.
Muromo mumwe chete wakanyorwa we pregabalin muvanhu wakabviswa muweti (92%) uye tsvina (<0.1%) pamusoro pemazuva mana. Urinary excretion zvigadzirwa zvaisanganisira zvinodhaka zvisina kuchinjwa (90% yedosi), N-Methylpregabalin (0.9%), nevamwe.
Single oral 75 kana 150 mg doses yakapiwa kuvanhu vane hutano yakapa peak urinary pregabalin concentrations ye151 kana 214 μg/mL, zvichiteerana, mumuenzaniso wekutanga we8-awa.
Pregabalin urine mazinga mu 57,542 zvienzaniso kubva kuvarwere vasingaperi vane 184 μg/mL.
Iyo PGB Pregabalin Test inopa mhedzisiro yakanaka apo pregabalin muweti inodarika 2,000 ng/mL.

