Testsealabs OXY Oxycodone Idanwo
Oxycodone: Alaye bọtini
Oxycodone jẹ opioid ologbele-sintetiki pẹlu ibajọra igbekalẹ si codeine. O jẹ iṣelọpọ nipasẹ iyipada thebaine, alkaloid kan ti a rii ninu poppy opium.
Gẹgẹbi gbogbo awọn agonists opiate, oxycodone pese iderun irora nipa ṣiṣe lori awọn olugba opioid ninu ọpa ẹhin, ọpọlọ, ati o ṣee ṣe taara ni awọn ara ti o kan. O ti paṣẹ fun iwọntunwọnsi si iderun irora giga labẹ awọn orukọ iṣowo ti a mọ daradara, pẹlu:
OxyContin®
Tylox®
Percodan®
Percocet®
Ni pataki, Tylox®, Percodan®, ati Percocet® ni awọn iwọn kekere ti oxycodone hydrochloride ni idapo pẹlu awọn analgesics miiran (fun apẹẹrẹ, acetaminophen tabi aspirin), lakoko ti OxyContin® ni oxycodone hydrochloride nikan ni fọọmu itusilẹ akoko.
Oxycodone metabolizes nipasẹ demethylation sinu oxymorphone ati noroxycodone. Fun iwọn lilo ẹnu 5mg kan, 33-61% ti yọ jade ninu ito wakati 24, pẹlu awọn eroja akọkọ jẹ:
Oogun ti ko yipada (13-19%)
Oogun ti a dapọ (7–29%)
Oksimorfoonu Asopọmọra (13–14%)
Ferese wiwa fun oxycodone ninu ito ni a nireti lati jọra si ti awọn opioids miiran (fun apẹẹrẹ, morphine).
Idanwo OXY Oxycodone mu abajade rere kan nigbati awọn ipele oxycodone ito kọja 100 ng/mL. Lọwọlọwọ, Abuse Abuse ati Isakoso Awọn Iṣẹ Ilera ti Ọpọlọ (SAMHSA) ko ti ṣe idasilẹ gige gige iboju ti a ṣeduro fun awọn apẹẹrẹ rere-oxycodone.

