Testsealabs OXY Oxycodone Gwajin
Oxycodone: Bayani mai mahimmanci
Oxycodone wani yanki ne na roba na roba tare da tsarin kamanni da codeine. Ana kera ta ta hanyar gyara thebaine, alkaloid da ake samu a cikin opium poppy.
Kamar duk opiate agonists, oxycodone yana ba da taimako na jin zafi ta hanyar yin aiki a kan masu karɓa na opioid a cikin kashin baya, kwakwalwa, da kuma yiwuwar kai tsaye a cikin kyallen takarda. An wajabta shi don matsakaita zuwa babban jin zafi a ƙarƙashin sanannun sunayen kasuwanci, gami da:
OxyContin®
Tylox®
Percodan®
Percocet®
Musamman ma, Tylox®, Percodan®, da Percocet® sun ƙunshi ƙananan allurai na oxycodone hydrochloride haɗe tare da sauran analgesics (misali, acetaminophen ko aspirin), yayin da OxyContin® ya ƙunshi oxycodone hydrochloride kawai a cikin hanyar sakin lokaci.
Oxycodone metabolizes ta hanyar demethylation zuwa oxymorphone da noroxycodone. Don kashi na baka na 5mg guda ɗaya, ana fitar da 33-61% a cikin fitsari na awa 24, tare da abubuwan farko sune:
Magunguna marasa canzawa (13-19%)
Magunguna masu haɗaka (7-29%)
Conjugated Oxymorphone (13-14%)
Ana sa ran taga gano oxycodone a cikin fitsari zai yi kama da na sauran opioids (misali, morphine).
Gwajin OXY Oxycodone yana haifar da sakamako mai kyau lokacin da matakan oxycodone na fitsari ya wuce 100 ng/mL. A halin yanzu, Hukumar Zagin Abu da Kula da Lafiyar Hauka (SAMHSA) ba ta kafa shawarar yankewar gwajin da aka yi ba don samfurori masu inganci na oxycodone.

