Testsealabs PGB Pregabalin Test
Pregabalin, analog na inhibitory neurotransmitter gamma-aminobutyric acid da kuma na gabapentin, an yi amfani dashi a asibiti tun 2002 azaman maganin analgesic, anticonvulsant, da anxiolytic wakili.
Ana ba da shi azaman magani kyauta a cikin capsules 25-300 MG don gudanar da baki. Magungunan manya yawanci suna cikin kewayon 50-200 MG sau uku a rana.
An kawar da kashi ɗaya na baki da aka yiwa lakabin pregabalin a cikin mutane a cikin fitsari (92%) da najasa (<0.1%) a tsawon kwanaki 4. Abubuwan fitar da fitsari sun haɗa da miyagun ƙwayoyi marasa canzawa (90% na kashi), N-Methylpregabalin (0.9%), da sauransu.
Magani na baka guda 75 ko 150 MG da aka ba mutane masu lafiya sun haifar da mafi girman adadin pregabalin na fitsari na 151 ko 214 μg/mL, bi da bi, a cikin samfurin sa'o'i 8 na farko.
Matakan fitsari na Pregabalin a cikin samfuran 57,542 daga marasa lafiya na ciwo na yau da kullun sun kai 184 μg/mL.
Gwajin PGB Pregabalin yana haifar da ingantaccen sakamako lokacin da matakin pregabalin a cikin fitsari ya wuce 2,000 ng/mL.

