Mayeso a Testsealabs OXY Oxycodone
Oxycodone: Zambiri
Oxycodone ndi opioid ya semi-synthetic yofanana ndi codeine. Amapangidwa ndi kusintha thebaine, alkaloid yomwe imapezeka mu opium poppy.
Monga ma opiate agonists onse, oxycodone imapereka mpumulo wopweteka pochita ma opioid receptors mumsana, ubongo, ndipo mwina mwachindunji m'magulu okhudzidwa. Amaperekedwa kuti athetse ululu wochepa mpaka wochepa pansi pa mayina odziwika bwino a malonda, kuphatikizapo:
OxyContin®
Tylox®
Percodan®
Percocet®
Makamaka, Tylox®, Percodan®, ndi Percocet® ali ndi timilingo tating'ono ta oxycodone hydrochloride kuphatikiza ndi mankhwala ena ochepetsa ululu (monga acetaminophen kapena aspirin), pomwe OxyContin® imakhala ndi oxycodone hydrochloride yokha mu mawonekedwe otulutsa nthawi.
Oxycodone imapangidwa kuchokera ku demethylation kukhala oxymorphone ndi noroxycodone. Pa mlingo umodzi wa 5mg pakamwa, 33-61% imatulutsidwa mumkodzo wa maola 24, ndipo zigawo zikuluzikulu ndizo:
Mankhwala osasinthidwa (13-19%)
Mankhwala osokoneza bongo (7-29%)
Conjugated oxymorphone (13-14%)
Zenera lozindikirira oxycodone mumkodzo likuyembekezeka kukhala lofanana ndi la ma opioid ena (mwachitsanzo, morphine).
Mayeso a OXY Oxycodone amapereka zotsatira zabwino pamene mikodzo ya oxycodone ya mkodzo iposa 100 ng/mL. Pakali pano, bungwe la Substance Abuse and Mental Health Services Administration (SAMHSA) silinakhazikitse njira yochepetsera yoyenelela ya zitsanzo za oxycodone-positive.

