Testsealabs PGB Pregabalin Test
Pregabalin, analogi wa inhibitory neurotransmitter gamma-aminobutyric acid komanso wa gabapentin, wakhala akugwiritsidwa ntchito kuchipatala kuyambira 2002 ngati mankhwala ochepetsa ululu, anticonvulsant, ndi anxiolytic agent.
Amaperekedwa ngati mankhwala aulere mu makapisozi a 25-300 mg kuti agwiritsidwe ntchito pakamwa. Mlingo wa akulu nthawi zambiri umakhala mkati mwa 50-200 mg katatu patsiku.
Mlingo umodzi wapakamwa wolembedwa wa pregabalin mwa anthu udachotsedwa mumkodzo (92%) ndi ndowe (<0.1%) pamasiku a 4. Mankhwala ochotsa mkodzo amaphatikizapo mankhwala osasinthika (90% a mlingo), N-Methylpregabalin (0.9%), ndi ena.
Mlingo umodzi wapakamwa wa 75 kapena 150 mg woperekedwa kwa anthu athanzi umatulutsa kuchuluka kwa mkodzo pregabalin wa 151 kapena 214 μg/mL, motsatana, m'chitsanzo choyambirira cha maola 8.
Mitsempha ya mkodzo wa Pregabalin mu zitsanzo za 57,542 kuchokera kwa odwala omwe ali ndi ululu wosatha pafupifupi 184 μg/mL.
Mayeso a PGB Pregabalin amapereka zotsatira zabwino pamene mlingo wa pregabalin mumkodzo umaposa 2,000 ng/mL.

