Testsealabs OXY Oxycodone Uvavanyo
Oxycodone: Ulwazi olungundoqo
I-Oxycodone yi-semi-synthetic opioid enesakhiwo esifana ne-codeine. Yenziwa ngokuguqula i-thebaine, ialkaloid efumaneka kwi-opium poppy.
Njengazo zonke i-opiate agonists, i-oxycodone inika isiqabu kwiintlungu ngokusebenza kwi-opioid receptors kwintambo yomgogodla, ingqondo, kwaye mhlawumbi ngokuthe ngqo kwizicubu ezichaphazelekayo. Imiselwe ukuthomalalisa okuphakathi ukuya kwintlungu ephezulu phantsi kwamagama arhweba awaziwayo, kubandakanywa:
OxyContin®
I-Tylox®
Percodan®
Percocet®
Ngokucacileyo, i-Tylox®, i-Percodan®, kunye ne-Percocet® ziqulethe iidosi ezincinci ze-oxycodone hydrochloride ezidityaniswe nezinye i-analgesics (umzekelo, i-acetaminophen okanye i-aspirin), ngelixa i-OxyContin® iqukethe kuphela i-oxycodone hydrochloride kwifom yokukhululwa kwexesha.
I-Oxycodone imetabolis nge-demethylation ibe yi-oxymorphone kunye ne-noroxycodone. Ngomlinganiselo omnye we-5mg yomlomo, i-33-61% ikhutshwe kumchamo weeyure ezingama-24, kunye neendawo eziphambili:
Iyeza elingatshintshwanga (13–19%)
Ichiza elidityanisiweyo (7–29%)
I-oxymorphone edityanisiweyo (13–14%)
Ifestile yokufunyanwa kwe-oxycodone kumchamo kulindeleke ukuba ifane neyezinye ii-opioids (umz., imorphine).
Uvavanyo lwe-OXY Oxycodone luvelisa iziphumo ezilungileyo xa amanqanaba e-oxycodone yomchamo edlula i-100 ng/mL. Kungoku nje, uLawulo lokuSetyenziswa gwenxa kweZiyobisi kunye noLawulo lweeNkonzo zeMpilo yeNgqondo (i-SAMHSA) alukaseka isindululo esicetyiswayo sokuhlolwa kwemizekelo ene-oxycodone-positive.

