Testsealabs PGB Pregabalin Test
I-Pregabalin, i-analog ye-inhibitory neurotransmitter gamma-aminobutyric acid kunye ne-gabapentin, isetyenziswe eklinikhi ukususela ngo-2002 njenge-analgesic, anticonvulsant, kunye ne-anxiolytic agent.
Inikezelwa njengechiza lasimahla kwii-capsules ze-25-300 mg zokulawulwa komlomo. Iidosi zabantu abadala ziqhelekile phakathi koluhlu lwe-50-200 mg kathathu yonke imihla.
Umthamo owodwa obhalwe ngomlomo we-pregabalin ebantwini upheliswe kumchamo (92%) kunye neefeces (<0.1%) kwixesha le-4-day. Iimveliso ze-Urinary excretion ziquka iziyobisi ezingatshintshiyo (90% yedosi), i-N-Methylpregabalin (0.9%), kunye nabanye.
Umlomo omnye we-75 okanye i-150 mg iidosi ezinikwe abantu abasempilweni zivelise i-peak urinary pregabalin concentrations ye-151 okanye i-214 μg/mL, ngokulandelanayo, kwi-specimen yokuqala ye-8 yeyure.
Amanqanaba omchamo we-Pregabalin kwiimpawu ze-57,542 ezivela kwizigulane ezibuhlungu ezingapheliyo zilinganiselwa kwi-184 μg / mL.
Uvavanyo lwe-PGB Pregabalin luvelisa umphumo omuhle xa izinga le-pregabalin kumchamo lidlula i-2,000 ng / mL.

