Testsealabs PGB Pregabalin Test
Pregabalin, analooga ah ee gamma-aminobutyric acid ee xannibaadda neurotransmitter iyo sidoo kale gabapentin, ayaa loo isticmaalay kiliinikada tan iyo 2002 sida xanuunka xanuunka, anticonvulsant, iyo wakiilka anxiolytic.
Waxaa lagu soo iibiyaa sida dawada bilaashka ah ee 25-300 mg kaabsal oo loogu talagalay maamulka afka. Qiyaasaha dadka waaweyn waxay caadi ahaan u dhexeeyaan 50-200 mg saddex jeer maalintii.
Hal dose oo afka ah oo lagu calaamadeeyay pregabalin ee bini'aadamka ayaa lagu tirtiray kaadida (92%) iyo saxarada (<0.1%) muddo 4-maalmood ah. Alaabooyinka kaadida ka soo baxa waxaa ka mid ahaa daroogo aan isbeddelin (90% qiyaasta), N-Methylpregabalin (0.9%), iyo kuwo kale.
Qiyaasta afka kaliya ee 75 ama 150 mg ee la siiyay bini'aadamka caafimaadka qaba waxay keeneen qiyaasta ugu sarreysa ee pregabalin kaadida ee 151 ama 214 μg/mL, siday u kala horreeyaan, muunadda 8-saac ee ugu horreysa.
Heerarka kaadida ee Pregabalin ee 57,542 shaybaarka bukaannada xanuunka daba dheeraada ayaa celcelis ahaan 184 μg/mL.
Tijaabada PGB Pregabalin waxay soo saartaa natiijo togan marka heerka pregabalin ee kaadidu uu dhaafo 2,000 ng/mL.

